Weight Loss + Dual Receptor

Tirzepatide

Sublingual Drops

Daily sublingual drops that activate two metabolic receptors simultaneously for blood sugar and weight control.

  • No Insurance Required

  • Ships From USA Pharmacy

  • Free Medical Consultation

  • No Subscription Required

  • Licensed Provider

  • Licensed Pharmacy

  • HIPAA Compliant

  • LegitScript Certified

Overview

Dual GIP/GLP-1 Agonist

Tirzepatide activates both GIP and GLP-1 receptors simultaneously, producing greater reductions in blood sugar and body weight than single-receptor agonism alone.

Mechanism of Action

Activates glucose-dependent insulinotropic polypeptide (GIP) and glucagon-like peptide-1 (GLP-1) receptors, increasing insulin secretion, decreasing glucagon secretion, increasing insulin sensitivity, and delaying gastric emptying

Sublingual Drops

Taken under the tongue once daily. Hold for 30 to 60 seconds before swallowing. Do not eat or drink for 15 minutes after administration.

Information presented here is for educational purposes only and not intended to replace or substitute guidance from a healthcare provider. Compounded medications are not FDA-approved nor evaluated by the FDA for safety, efficacy, or quality.

Benefits

Dual Receptor Action

Activates GIP and GLP-1 pathways together, driving fat metabolism, appetite suppression, and blood sugar control beyond what GLP-1 alone achieves.

Appetite Control

Mimics two postprandial hormones to signal the brain to reduce hunger and slow digestion for extended satiety.

Blood Sugar Regulation

Stimulates insulin secretion, suppresses glucagon, and slows gastric emptying through two complementary mechanisms.

Needle-Free

A convenient daily alternative to weekly injectable tirzepatide for patients who prefer an oral route of administration.

Individual results may vary. Benefits described are based on clinical and pharmacological evidence and do not constitute a guarantee of treatment outcomes. All treatment requires evaluation and approval by a licensed provider.

Simple. Medical. Personalized.

Medical intake

Answer a few online questions about your health history, lifestyle, & goals. No clinic visits required.

Provider evaluation

A licensed medical provider reviews your intake to determine the safest, personalized treatment.

Personalized plan

Custom treatment plan built around your unique health needs, goals, medical history, & biology.

Ongoing support

Stay connected with your care team for follow-ups, adjustments, & expert answers 100% online.

FAQs

What is Tirzepatide Sublingual Drops?

Tirzepatide Sublingual Drops is a prescription therapy used for metabolic and weight management support.

Who should use Tirzepatide Sublingual Drops?

Patients seeking support for metabolic and weight management support may qualify after evaluation by a licensed provider.

Does Tirzepatide Sublingual Drops require a prescription?

Yes. This compounded medication is dispensed by Strive Pharmacy pursuant to a valid prescription from a licensed provider following a telemedicine evaluation.

What are the possible side effects?

Common side effects include nausea, vomiting, diarrhea, constipation, and abdominal discomfort, particularly during the first few weeks as your body adjusts. These typically improve with continued use. Worsening of diabetic retinopathy has been reported — patients with a history of retinopathy should be monitored closely by their provider. Pancreatitis has been reported with this drug class — discontinue use and contact your provider immediately if you experience persistent, severe abdominal pain. In animal studies, GIP/GLP-1 receptor agonists have been associated with thyroid C-cell tumors; the relevance to humans is not established, but this medication is contraindicated in patients with a personal or family history of medullary thyroid carcinoma or MEN 2.

Who Should Not Use Tirzepatide Sublingual Drops?

Not for use in patients with a personal or family history of medullary thyroid carcinoma or MEN 2. Not recommended during pregnancy. Do not use alongside other GLP-1 or GIP receptor agonists.

Are there any drug interactions?

Tirzepatide may slow gastric emptying and affect the absorption timing of other oral medications. Do not combine with other GLP-1 or GIP agonists. Disclose all medications to your provider.

Is Tirzepatide Sublingual Drops safe if I have a pre-existing medical condition?

Not recommended for patients with severe GI disease, active pancreatitis, or significant renal impairment. Patients with diabetic retinopathy should be monitored closely. Full provider review is required.

Contact Us

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Hours

Monday–Saturday, 10am–8pm ET

Text or Call

Hours

Monday–Saturday, 10am–8pm ET

Start Your Journey

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Physician-supervised. Delivered to your door.

No clinic visits required.

  • Licensed Provider

  • Licensed Pharmacy

  • HIPAA Compliant

  • LegitScript Certified

The information and clinical services described on this website are for educational and informational purposes only and are not intended to diagnose, treat, cure, or prevent any disease. All treatments require evaluation and approval by a licensed healthcare provider through a telemedicine consultation. Treatment approval is not guaranteed. Individual results may vary, and treatments may carry risks and side effects. Certain compounded medications, wellness treatments, or off-label uses may not be evaluated by the U.S. Food and Drug Administration (FDA) for safety, effectiveness, or quality unless explicitly stated. Testosterone Shots provides telehealth consultations, clinical review, care coordination, lab-related services, membership services, and ongoing treatment management. Testosterone Shots is not a pharmacy and does not manufacture, compound, dispense, sell, handle, warehouse, ship, or collect payment for prescription medication. Testosterone Shots collects payment only for consultations, clinical review, care coordination, lab-related services, membership services, and other non-pharmacy services. If treatment is approved, your prescription may be sent to a licensed pharmacy partner. The pharmacy contacts you directly to complete medication payment and shipping. Services are provided by licensed physicians, nurse practitioners, and/or other licensed healthcare providers in states where they are authorized to practice. This service is not intended for medical emergencies. If you are experiencing an emergency, call 911 or seek immediate medical care. We take reasonable measures to protect personal health information in accordance with applicable privacy laws, including HIPAA. By using this website or its services, you agree to our Terms of Service, Privacy Policy, Notice of Privacy Practices, Telehealth Consent, and Important Safety Information. You must be 18 years of age or older to use this service.